SHARP Paula Luiz (US),ШАРП Паула Луиз (US),STIVENSON Tomas Martin (US),СТИВЕНСОН Томас Мартин (US),DEPRE Nikolya Rajan (US),ДЕПРЕ Николя Райан (US),REDDI Ravisekkhara P. (IN),РЕДДИ Рависекхара П. (IN)
申请号：
RU2016127518
公开号：
RU0002703460C1
申请日:
2014.12.09
申请国别(地区):
RU
年份:
2019
代理人:
摘要：
FIELD: chemistry.SUBSTANCE: invention relates to a novel compound of formula 1 or a salt thereof. In the compound of formula 11 -Y1= Y2-Y3= Y4-, including nitrogen atom, to which are connected as Y1, and Y4, selected fromZ is O or S； each R1 independently represents hydrogen, halogen, cyano, nitro, CHO, C(= O)NH2, SO2NH2, C1-C4alkyl, C2-C4alkenyl, C2-C4alkynyl, C1-C4haloalkyl, C3-C6cycloalkyl, C2-C6alkylcarbonyl, C2-C6alkoxycarbonyl, C1-C4alkoxy, C1-C4haloalkoxy, C2-C6cyanoalkoxy, SOnR1A, Si (CH3)3, C (= (NOH) CH3 or B (-OC (R1B)2C (R1B)2O-)； or a phenyl ring optionally substituted with not more than 5 substitutes independently selected from R1C； or 5- or 6-member heteroaromatic ring containing ring members selected from carbon atoms and not more than 4 heteroatoms independently selected from at most 2 O atoms, not more than 2 S atoms and not more than 4 N atoms, wherein each ring is optionally substituted with not more than 3 substitutes independently selected from R1C by ring members, which are carbon atoms, and R1D by ring members, which are nitrogen atoms； R2 is halogen, cyano, nitro, C1-C4alkoxy, C1-C4alkyl, C2-C6alkynyl or C1-C4haloalkyl； m is 0, 1, 2 or 3； each R3 independently represents halogen, cyano, hydroxy, nitro, CHO, C(= O)NH2, C(= S)NH2, C1-C4alkyl, C2-C4alkenyl, C2-C4alkynyl, C1-C4haloalkyl, C2-C6alkylcarbonyl, C1-C4alkoxy, C1-C4haloalkoxy, C2-C4alkylcarbonyloxy, C≡CSi (CH3)3, C (= O) N (R3A) (R3B), C (= NOR3C) H, C (= NR3D) H, SOnR3E； or a phenyl ring optionally substituted with not more than 5 substitutes independently selected from R3F； or 5- or 6-member heteroaromatic ring containing ring members selected from carbon atoms and not more than 4 heteroatoms independently selected from at most 2 O atoms, not more than 2 S atoms and not more than 4 N atoms, wherein each ring is optionally substituted with not more than 3 substitutes independently selected from R3F by ring members, which are carbon atoms, and R3G by ring members, which are nitrogen at
