Gonzalo Hernández Herrero,Victor Rubio Royo,Neftalí García Domínguez,Gonzalo Canal Mori,Nicolas Tesson
申请号:
US15777132
公开号:
US20180344854A1
申请日:
2016.11.18
申请国别(地区):
US
年份:
2018
代理人:
摘要:
The invention relates to a stable supersaturated aqueous solution comprising bilastine and an selected from glutaric acid, citric acid, α-cetoglutaric acid, tartaric acid, acetic acid, propionic acid and mixtures thereof and to its use in the treatment and/or prevention of conditions mediated by H1 histamine receptor, such as allergic disorders or diseases. The invention also relates to the use of the above organic carboxylic acids to increase the aqueous solubility of bilastine.