Matthias Witschel,Frank Stelzer,Johannes Hutzler,Tao Qu,Thomas Mietzner,Klaus Kreuz,Klaus Grossmann,Raphael Aponte,Hans Wolfgang Hoeffken,Frederick Calo,Thomas Ehrhardt,Anja Simon,Liliana Parra Rapado
申请号:
US14405942
公开号:
US09480259B2
申请日:
2013.05.29
申请国别(地区):
US
年份:
2016
代理人:
摘要:
The present invention relates to a pyrazolopyran of the general formula I wherein the variables are defined according to the description, including a tautomer, salt, cleavable prodrug, or mixtures thereof, in particular to said pyrazolopyran for use as a medicament and/or an inhibitor of the enzyme serinehydroxymethyltransferase (SHMT). The invention also relates to a process the preparation of a pyrazolopyran of the formula I, to compositions comprising said compound and processes for the preparation of these compositions. Further it relates to use of the pyrazolopyran of formula I as an herbicide as well as to a method of controlling undesired vegetation.