您的位置: 首页 > 农业专利 > 详情页

SULFONAMIDE INHIBITORS OF HIV-ASPARTYL PROTEASE, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SULFONAMIDES AND PROCESS FOR PREPARING THEM
专利权人:
VERTEX PHARMACEUTICALS INCORPORATED; CAMBRIDGE
发明人:
BHISETTI, GOVINDA RAO,MURCKO, MARK A.,TUNG, ROGER D.
申请号:
HU9500685
公开号:
HU228198B1
申请日:
1993.09.07
申请国别(地区):
HU
年份:
2013
代理人:
摘要:
The present invention relates to a novel class of sulfonamides which are aspartyl protease inhibitors, of formula (I). In one embodiment, this invention relates to a novel class of HIV aspartyl protease inhibitors characterized by specific structural and physicochemical features. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibiting HIV-1 and HIV-2 protease activity and consequently, may be advantageously used as antiviral agents against the HIV-1 and HIV-2 viruses. This invention also relates to methods for inhibiting the activity of HIV aspartyl protease using the compounds of this invention and methods for screening compounds for anti-HIV activity. <;CHEM>;
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充