CONDE-KNAPE, KARIN,DANHO, WALEED,EHRLICH, GEORGE,FOTOUHI, NADER,FRY, DAVID C.,KHAN, WAJIHA,KONKAR, ANISH,RONDINONE, CRISTINA MARTHA,SWISTOK, JOSEPH,TAUB, REBECCA ANNE,TILLEY, JEFFERSON W.
申请号:
AT06830133
公开号:
AT549350T
申请日:
2006.11.27
申请国别(地区):
AT
年份:
2012
代理人:
摘要:
Provided herein are neuropeptide-2 receptor agonists of the formula (I): as well as pharmaceutically acceptable salts, derivatives and fragments thereof, wherein the substituents are as those disclosed in the specification. X is 4-oxo-6-(1-piperazinyl)-3(4H)-quinazoline-acetic acid (Pqa). These compounds, and the pharmaceutical compositions containing them, are useful for the treatment of diseases such as, for example, obesity and diabetes.