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具有環狀構造的化合物
专利权人:
DAIICHI SANKYO COMPANY; LIMITED
发明人:
TANIGUCHI, TORU,谷口亨,谷口亨,IWAMOTO, OSAMU,岩本理,岩本理,SAITO, KEIJI,斋藤啓志,齋藤啓志,NAKAJIMA, KATSUYOSHI,中岛胜义,中島勝義,OGAWA, YASUYUKI,小川泰之,小川泰之,KURIKAWA, NOBUYA,栗川伸也,栗川伸也,NAGATA, SEIKO,长田圣子,長田聖子,ITO, KAORI,伊藤香织,伊藤香織,K
申请号:
TW107132188
公开号:
TW201920153A
申请日:
2018.09.13
申请国别(地区):
TW
年份:
2019
代理人:
摘要:
The present invention addresses the problem of providing a compound having an anti-inflammatory effect, a pharmacologically acceptable salt thereof, etc. The means for solution according to the present invention is a compound represented by general formula (I) or a pharmacologically acceptable salt thereof. (The symbols in the formula are defined as follows. A: benzene, etc.; E: -CH2-, etc.; G: a five-membered aromatic heterocycle, etc.; X: cyclohexane, etc.; J: a five-membered aromatic heterocycle, etc.; Y: a phenyl group, etc.; R1, R2, and R3: a halogen atom, etc.; R4: a C1-6 alkyl group, etc.; R5: a hydrogen atom, etc.; R6a, R6b, R6c, and R6d: a hydrogen atom, etc.; R7: a hydrogen atom, etc.; R8: a hydrogen atom, etc.; n1, n2, n3: 1, etc.).本發明之課題,係提供具有抗炎症作用的化合物、其藥理上可容許的鹽等。本發明之解決手段,係通式(1)之化合物或其藥理上可容許的鹽。[式中之記號係定義於下。A:苯等;E:-CH2-等;G:5員芳香族雜環等;X:環己烷等;J:5員芳香族雜環等;Y:苯基等;R1、R2、R3:鹵素原子等;R4:C1-C6烷基等;R5:氫原子等;R6a、R6b、R6c、R6d:氫原子等;R7:氫原子等;R8:氫原子等;n1、n2、n3:1等]
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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