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Chiral diacylhydrazine ligands to modulate exogenous genetic expression through the ecdysone receptor complex
- 专利权人:
- Intrexon Corporation
- 发明人:
- HORMANN, Robert,LI, Bing
- 申请号:
- ES08754763
- 公开号:
- ES2672513T3
- 申请日:
- 2008.05.29
- 申请国别(地区):
- ES
- 年份:
- 2018
- 代理人:
- 摘要:
- A compound selected from the group consisting of: (R) -3,5-Dimethyl-benzoic acid N- (1-tert-butyl-butyl) -N '- (2-ethyl-3-methoxybenzoyl) -hydrazide; (R) -3,5-Dimethyl-benzoic acid N'-benzoyl-N- (1-tert-butyl-butyl) -hydrazide; (R) -3,5-5 dimethyl-benzoic acid N- (1-tert-butyl-butyl) -N '- (2-methyl-benzoyl) -hydrazide; (R) -3,5-Dimethyl-benzoic acid N- (1-tert-butyl-butyl) -N '- (2-fluoro-benzoyl) -hydrazide; (R) -3,5-Dimethyl-benzoic acid N '- (2-bromo-benzoyl) -N- (1-tert-butyl-butyl) -hydrazide; (R) -3,5-Dimethyl-benzoic acid N- (1-tert-butyl-butyl) -N '- (3-methyl-benzoyl) -hydrazide; (R) -3,5-Dimethyl-benzoic acid N- (1-tert-butyl-butyl) -N '- (4-methyl-benzoyl) -hydrazide; (R) -3,5-Dimethyl-benzoic acid N- (1-tert-butyl-butyl) -N '- (2-chloro-pyridine-3-carbonyl) -hydrazide; (R) -3,5-Dimethyl-benzoic acid N- (1-tert-butyl-butyl) -N '- (6-chloro-pyridine-3-carbonyl) -hydrazide; and N- (1-tert-butyl-butyl) -N'- (3-methoxy-2-methyl-benzoyl) -hydrazide (R) -3,5-dimethyl-benzoic acid, or a pharmaceutically acceptable salt of the same.Un compuesto seleccionado del grupo que consiste de: N-(1-tert-butil-butil)-N'-(2-etil-3-metoxibenzoil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; N'-benzoil-N-(1-tert-butil-butil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; N-(1-tert-butil-butil)-N'-(2-metil-benzoil)-hidrazida de ácido (R)-3,5-5 dimetil-benzoico; N-(1-tert-butil-butil)-N'-(2-fluoro-benzoil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; N'-(2-bromo-benzoil)-N-(1-tert-butil-butil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; N-(1-tert-butil-butil)-N'-(3-metil-benzoil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; N-(1-tert-butil-butil)-N'-(4-metil-benzoil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; N-(1-tert-butil-butil)-N'-(2-cloro-piridina-3-carbonil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; N-(1-tert-butil-butil)-N'-(6-cloro-piridina-3-carbonil)-hidrazida de ácido (R)-3,5-dimetil-benzoico; y N-(1-tert-butil-butil)-N'- (3-metoxi-2-metil-benzoil)-hidrazida de á
- 来源网站:
- 中国工程科技知识中心
- 来源网址:
- http://www.ckcest.cn/home/