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compound use of a compound and pharmaceutical composition
专利权人:
ICAHN SCHOOL OF MEDICINE AT MOUNT SINAI
发明人:
David Kastrinsky,Michael Ohlmeyer
申请号:
BR112015019818
公开号:
BR112015019818A2
申请日:
2014.02.19
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
1/1 summary "compound, use of a compound, and pharmaceutical composition" tricyclic chemical modulators of fox transcription factor proteins are described. The compounds are used to treat cancer, age-onset proteotoxicity, stress-induced depression, inflammation and acne. the compounds are of the following genera and the like: het het het het yyy, and wherein het is an aromatic heterocyclic ring and y is an attachment point of several side chains and rings . An example of such a compound is 4-chloro-n- (3- (10,11-dihydro-5h-benzo [b] pyrido [2,3-f] azepin-5-yl) propyl) benzenesulfonamide : nn cl osnoh.1 / 1 resumo “composto, uso de um composto, e, composiã‡ãƒo farmacãšuticaâ€� sã£o descritos moduladores quã­micos tricã­clicos das proteã­nas do fator de transcriã§ã£o foxo. os compostos sã£o usados para tratar cã¢ncer, proteotoxicidade com inã­cio de aã§ã£o por idade, depressã£o induzida por estresse, inflamaã§ã£o e acne. os compostos sã£o dos seguintes gãªneros e similares: het het het het y y y , e em que het ã© um anel heterocã­clico aromã¡tico e y ã© um ponto de anexaã§ã£o de vã¡rias cadeias laterais e anã©is. um exemplo de um composto como este ã© 4-cloro-n-(3-(10,11-di-hidro-5h-benzo[b]pirido[2,3-f]azepin-5- il)propil)benzenossulfonamida: n n cl o s n o h .
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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