ANDREW DUNCAN SATTERFIELD,THOMAS MARTIN STEVENSON,MATTHEW JAMES CAMPBELL
申请号：
ARP160101388
公开号：
AR104618A1
申请日:
2016.05.12
申请国别(地区):
AR
年份:
2017
代理人:
摘要：
Claim 1: a compound (1) selected from the formula,N-sulfur oxide, stereoisomers and their salts, Q1 is phenyl or benzene ring, or nafterenio ring system； each ring or ring system can be replaced by up to five independent alternatives r8313；Or a completely unsaturated 5-6-member heteroaromatic ring or 8-10 member heteroaromatic bicyclic ring system； each ring or ring system contains ring members selected from carbon atoms and 1-4 selected heteroatoms, but no more than 2 O atoms, Up to two S atoms and up to four N atoms, of which up to three carbon ring members independently choose C (= O) and C (= s),The sulfur atom in the ring is independent of S (= O) 751222 (= n831222) 7515e；Each ring or ring system can be replaced by up to five substitutes selected independently from r8313. These substitutes come from the ring part of carbon atom, which is selected as r83044 in the ring part of nitrogen atom； Q2 is a phenyl ring or nataleni ring system； each ring or ring system. 1. It can be replaced by up to 5 substitutes selected by independent R1；Or a completely unsaturated 5-6-member heteroaromatic ring or 8-10 member heteroaromatic bicyclic ring system； each ring or ring system contains ring members selected from carbon atoms and 1-4 selected heteroatoms, but no more than 2 O atoms, Up to two S atoms and up to four N atoms, of which up to three carbon ring members independently choose C (= O) and C (= s),The sulfur atom in the ring is independent of S (= O) 751222 (= n831222) 7515e；each ring or ring system is optionally substituted with up to 5 substituents independently selected from R¹¹ in ring members that are carbon atoms and selected from R¹² in ring members that are nitrogen atoms； R¹ and R² are each independently H, halogen, hydroxyl or C₁₋₄ alkyl；Y is O, S or NR¹⁵；A is a saturated, partially or completely unsaturated chain consisting of two to four atoms selected from a maximum of four carbon atoms, a maximum of one O atom, a maximum of one s atom, and a maximum of t
