PEGG, NEIL ANTHONY,TADDEI, DAVID MICHEL ADRIEN,SHANNON, JONATHAN,PAOLETTA, SILVIA,QIN, TING,HARBOTTLE, GARETH
申请号:
CA3039643
公开号:
CA3039643A1
申请日:
2017.10.18
申请国别(地区):
CA
年份:
2018
代理人:
摘要:
A compound which is a benzimidazole of formula (I): wherein X is a 5-membered heteroaryl group selected from the following: or a pharmaceutically acceptable salt thereof. The compound has activity in modulating the activity of p300 and/or CBP and is used to treat cancer, particularly prostate cancer.