您的位置: 首页 > 农业专利 > 详情页

compounds and their use
专利权人:
Orchid Chemicals and Pharmaceuticals Ltd.
发明人:
Aravind Appu,Gopalan Balasubramanian,Hariharan Periasamy,Maneesh Paul-Satyaseela,Senthilkumar Udayampalayam Palanisamy,Senthilnathan Manickam,Shridhar Narayanan
申请号:
BR112013012735
公开号:
BR112013012735A2
申请日:
2011.11.25
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
compounds and their use. The present invention relates to compounds and their use in the treatment of infections. The compound of formula (I), its derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, solvates, pharmaceutically acceptable salts and pharmaceutical compositions described herein are also useful as β-lactamase inhibitors, which restore or increase the antibiotic spectrum of a suitable antibiotic agent. The compounds of formula (I) act as β-lactamase inhibitors. These compounds restore / potentiate the activities of β-lactam antibiotics against carbapenemases. Such compounds find use in a diagnostic method for detecting β-lactamases.compostos e seu uso. a presente invenção refere-se a compostos e seu uso no tratamento de infecções. o composto da fórmula (i), seus derivados, análogos, formas tautoméricas, estereoisômeros, polimorfos, solvatos, sais farmaceuticamente aceitáveis e composições farmacêuticas descritos aqui também são úteis como inibidores <;225>;-lactamase, os quais restauram ou aumentam o espectro antibiótico de um agente antibiótico adequado. os compostos da fórmula (i) atuam como inibidores de <;225>;-lactamases. esses compostos restauram/potencializam as atividades de antibióticos de <;225>;-lactamas contra carbapenemases. esses compostos encontram uso em método de diagnóstico para detectar <;225>;-lactamases.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充