BERNARDES, GONCALO,RODRIGUES, TIAGO,CONDE, JOAO,BAKER, CHARLOTTE
申请号：
CA3075981
公开号：
CA3075981A1
申请日:
2018.09.14
申请国别(地区):
CA
年份:
2019
代理人:
摘要：
This invention relates to the finding that Piperlongumine compounds, such as Piperlongumine and analogues, derivatives and prodrugs thereof, are reversible, allosteric antagonists of transient receptor potential vanilloid 2 channel (TRPV2). Methods of treatment of conditions that are characterised by TRPV2 expression using Piperlongumine compounds and Piperlongumine compounds for use in such treatments are provided
