GOMME, Justin,DI GIORGIO, Patrick,MATTEI, Patrizio,HERT, Jérôme,HUNZIKER, Daniel,SCHMITZ, Petra,RUDOLPH, Markus
申请号：
CR20190423
公开号：
CR20190423A
申请日:
2018.03.13
申请国别(地区):
CR
年份:
2019
代理人:
摘要：
The invention provides a new compound. In the general formula (I), R1, R2, y, x, W, m and N are the compounds defined in this document, including the compound and the method for using the compound. The invention provides a new compound. The general formula (I) where R1 is selected from the alternatives. Phenyl，pyridinyl or thiophenyl，R2 is selected from optimonally substituted aminosulfonylphenyl，aminosulfonylpyridinyl，aminosulpholthiophenyl or aminosulphyalthiazyll，x is nitrogen or carbon，and is a linking group，Z is a direct bond or a linking group，M=0-5，n=0-5 with the provision that M+N is 2-5，Compositions including the compounds and the use of the compounds in the treatment or prophylaxis of object conditions.La invención proporciona nuevos compuestos que tienen la fórmula general (I)(I) en la que R1, R2, Y, X, W, m y n son como se definen en el presente documento, composiciones que incluyen los compuestos y métodos de uso de los compuestos.The invention provides novel compounds having the general formula (I) wherein R1 is selected from substituted phenyl, pyridinyl or thiophenyl, R2 is selected from optionally substituted aminosulphonylphenyl, aminosulphonylpyridinyl, aminosulphonylthiophenyl or aminosulphonylthiazolyl, X is nitrogen or carbon, Y is a linking group, Z is a direct bond or a linking group, m = 0-5, n = 0-5 with the proviso that m+n is 2-5, compositions including the compounds and the use of the compounds in the treatment or prophylaxis of ocular conditions.
