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PHARMACEUTICALLY ACCEPTABLE SALTS OF 2-{ 4-[(3S)-PIPERIDIN-3- YL]PHENYL} -2H-INDAZOLE-7-CARBOXAMIDE
- 专利权人:
- MERCK SHARP & DOHME LIMITED
- 发明人:
- FOLEY, JENNIFER, R,WILSON, ROBERT DARRIN
- 申请号:
- NZ58667509
- 公开号:
- NZ586675A
- 申请日:
- 2009.01.08
- 申请国别(地区):
- NZ
- 年份:
- 2012
- 代理人:
- 摘要:
- Disclosed are compounds selected from: (3S)-3-{ 4-[7-(Aminocarbonyl)-2H-indazol-2-yl]phenyl} piperidinium 4-methylbenzenesulfonate (3S)-3-{ 4-[7-(Aminocarbonyl)-2H-indazol-2-yl]phenyl} piperidinium sulfate (3S)-3-{ 4-[7-(Aminocarbonyl)-2H-indazol-2-yl]phenyl} piperidinium benzenesulfate (3S)-3-{ 4-[7-(Aminocarbonyl)-2H-indazol-2-yl]phenyl} piperidinium fumarate (3S)-3-{ 4-[7-(Aminocarbonyl)-2H-indazol-2-yl]phenyl} piperidinium succinate (3S)-3-{ 4-[7-(Aminocarbonyl)-2H-indazol-2-yl]phenyl} piperidinium 4-methylbenzenesulfonate monohydrate. The compounds are used to treat cancer, inflammatory diseases, reperfusion injuries, ischemic conditions, stroke, renal failure, cardiovascular diseases, vascular diseases other than cardiovascular diseases, diabetes, neurodegenerative diseases, retroviral infection, retinal damage or skin senescence and UV induced skin damage.
- 来源网站:
- 中国工程科技知识中心
- 来源网址:
- http://www.ckcest.cn/home/