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COMPOUNDS HAVING CRTH2 ANTAGONIST ACTIVITY
专利权人:
ATOPIX THERAPEUTICS LIMITED
发明人:
ARMER, RICHARD EDWARD,PETTIPHER, ERIC ROY,WHITTAKER, MARK,WYNNE, GRAHAM, MICHAEL,VILE, JULIA,SCHROER, FRANK
申请号:
MYPI 2010003390
公开号:
MY155133A
申请日:
2009.01.19
申请国别(地区):
MY
年份:
2015
代理人:
摘要:
COMPOUNDS OF GENERAL FORMULA (I) WHEREIN W IS CHLORO OR FLUORO; R1 IS PHENYL OPTIONALLY SUBSTITUTED WITH ONE OR MORE SUBSTITUENTS SELECTED FROM HALO,-CN, -C1-C6 ALKYL, -SOR3, -SO2R3, -SO2N(R2)2, -N(R2)2, -NR2C(O)R3, -CO2R2, -CONR2R3, -NO2, -OR2, -SR2, -O(CH2)pOR2, AND -O(CH2)pO(CH2)qOR2 WHEREIN EACH R2 IS INDEPENDENTLY HYDROGEN, -C1-C6 ALKYL, -C3-C8 CYCLOALKYL, ARYL OR HETEROARYL; EACH R3 IS INDEPENDENTLY, -C1-C6 ALKYL, -C3-C8 CYCLOALKYL, ARYL OR HETEROARYL; p AND q ARE EACH INDEPENDENTLY AN INTEGER FROM 1 TO 3; AND THEIR PHARMACEUTICALLY ACCEPTABLE SALTS, HYDRATES, SOLVATES, COMPLEXES OR PRODRUGS ARE USEFUL IN ORALLY ADMINISTRABLE COMPOSITIONS FOR THE TREATMENT OF ALLERGIC DISEASES SUCH AS ASTHMA, ALLERGIC RHINITIS AND ATOPIC DERMATITIS.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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