MATTHIAS NETTEKOVEN,MARK ROGERS-EVANS,CATERINA BISSANTZ,UWE GRETHER,ATSUSHI KIMBARA,JEAN ADAM,STEPHAN MICHEL - ROEVER
申请号：
ARP120104159
公开号：
AR088663A1
申请日:
2012.11.06
申请国别(地区):
AR
年份:
2014
代理人:
摘要：
1. Claim 1: a compound of formula (1), wherein: A is asphalt, nitrous hydroxide, ch8322； (c) (o)-C (O) --SO₂- or is absent； R¹ is hydrogen, alkyl, haloalkyl, hydroxy, alkoxy, haloalkoxy, phenyl, halophenyl, alkoxyphenyl, haloalkylphenyl, haloalkoxyphenyl, (halo) (haloalkyl) phenyl, cyanophenyl, hydroxyalkoxyphenyl, alkylsulfonylphenyl, alkylsulfonylaminophenyl, cycloalkylalkyl, cycloalkylalkyl, cycloalkylalkyl, cycloalkyloxylalkyl, cycloalkylalkyl ) (alkyl) [1,2,4] tri-azolyl, (halo) (dialkylamino) pyridinyl, (alkyl) (oxy) pyridinyl, nitro-benzo [1,2,5] oxadiazolylaminopyridinyl, heterocyclyl, alkylheterocyclyl, hydroxyheterocyclyl, alkylheterocyclyl , heteroaryl, haloheteroaryl, alkylheteroaryl, cycloalkylheteroaryl or haloalkylheteroaryl,1. Isocyclic propene is a carbon ring composed of 3 to 8 members, containing at least one nitrogen or oxygen atom； heteromorphism is: pyridine, pyridine, pyridine, oxadiazolo, furan, tetratoluene or trimethylene； R2 is halogen, NR: r8308o-or83099；one of R³ and R⁴ is hydrogen or alkyl and the other is alkyl or cycloalkyl； or R³ and R⁴ together with the nitrogen atom to which they are attached form a substituted heterocyclyl or heterocyclyl, said heterocyclyl is morpholinyl, piperidinyl, piperazinyl, pyrrolidinyl, 2-oxa-6-azaspiro [3.3] heptyl, azetidinyl, thiazolidinyl, thiomorinyl, thiomorinyl, thiomorinyl dioxothiomorpholinyl, oxazepanyl, 2-oxa-6-azaespiro [3.4] octyl, 6-oxa-1-azaspiro [3.3] heptyl, 2-oxa-5-azaespiro [3.4] -octyl, isoxazolidinyl, aziridinyl, dioxoisothiazolidinyl or oxydiopyridinyl substituted heterocyclyl is a heterocyclyl substituted one to four times by substituents independently selected from alkyl,Halogen, hydroxyl, alcoxi, hydroxil, hydroxilo, carboxilo, ALCOXY codique, Ciano, autorimino, dialcamino, alcoholamino, lcarbonial (rent)1. Phenyl, alcoxicarbon, carbamate, alkylpicolinate and alkyllisoxazolilo； r83099 is tar, cyclopentadiene, cyclopropylic acid, halotars or oxetanilo； or a salt or ester acceptable
