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DERIVATIVES OF INDOLE-2-CARBOXAMIDES AND OF AZAINDOLE-2-CARBOXAMIDES SUBSTITUTED WITH A SILANYL GROUP, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
专利权人:
SANOFI-AVENTIS
发明人:
LAURENT DUBOIS,YANNICK EVANNO,ANDRÉ MALANDA
申请号:
MYPI 2010003446
公开号:
MY150289A
申请日:
2009.01.20
申请国别(地区):
MY
年份:
2013
代理人:
摘要:
THE INVENTION RELATES TO COMPOUNDS OF THE GENERAL FORMULA (I) IN WHICH: G₁, G₂, G₃ ET G₄ ARE INDEPENDENT FROM ONE ANOTHER, A C-X GROUP OR A NITROGEN ATOM; ONE OF G₁, G₂, G₃ AND G₄ AND AT MOST ONE OF G₁, G₂, G₃ AND G₄IS A C-X GROUP IN WHICH X IS A -Si(X₁)(X₂)(X₃) GROUP; N IS 0, 1, 2 OR 3; Y IS AN OPTIONALLY SUBSTITUTED ARYL OR HETEROARYL; ZI, Z2, Z3, Z4 ARE INDEPENDENT FROM ONE ANOTHER, A NITROGEN ATOM OR A C(R₆) GROUP, AT LEAST ONE BEING A NITROGEN ATOM AND AT LEAST ONE BEING A C(R₆) GROUP; Z IS CYCLIC AMINO OR ACYCLIC AMINO; SAID COMPOUNDS CAN BE IN THE STATE OF A BASE OR AN ADDITION SALT TO AN ACID, AS WELL AS IN THE HYDRATE OR SOLVATE STATE. THE INVENTION ALSO RELATES TO A METHOD FOR PREPARING THE SAME AND TO THE THERAPEUTIC USE THEREOF.
来源网站:
中国工程科技知识中心
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http://www.ckcest.cn/home/

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