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morpholine and 1,4-oxazepane amides as agonists of the somatostatin 4 receptor subtype (sstr4)
专利权人:
BOEHRINGER INGELHEIM INTERNATIONAL GMBH
发明人:
IAIN LINGARD,KLAUS RUDOLF,MARCO FERRARA,RICCARDO GIOVANNINI,ROCCO MAZZAFERRO
申请号:
BR112017009595
公开号:
BR112017009595A2
申请日:
2015.11.12
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
The present invention relates to morpholine and 1,4-oxazepane amide derivatives of general formula (I) which are agonists of the somatostatin 4 receptor subtype (sstr4) useful for preventing or treating medical disorders related to the disease. sstr4. furthermore, the invention relates to processes for the preparation of pharmaceutical compositions as well as processes for the manufacture of compounds according to the invention.a presente invenção refere-se aos derivados de morfolina e 1,4-oxazepano amida de fórmula geral (i), os quais são agonistas do subtipo de receptor de somatostatina 4 (sstr4), úteis para prevenir ou tratar os distúrbios médicos relacionadas com o sstr4. além disso, a invenção refere-se aos processos para a preparação de composições farmacêuticas, assim como aos processos para a fabricação dos compostos de acordo com a invenção.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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