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INHIBITORS OF SERINE PROTEASES, PARTICULARLY HCV NS3-NS4A PROTEASE
专利权人:
VERTEX PHARMACEUTICALS INCORPORATED
发明人:
ROBERT B. PERNI,JOHN J. COURT,SHAWN D. BRITT,JANOS PITLIK,JOHN H. VAN DRIE
申请号:
MYPI 20043610
公开号:
MY148123A
申请日:
2004.09.06
申请国别(地区):
MY
年份:
2013
代理人:
摘要:
THE PRESENT INVENTION RELATES TO COMPOUNDS THAT INHIBIT SERINE PROTEASE ACTIVITY, PARTICULARLY THE ACTIVITY OF HEPATITIS C VIRUS NS3-NS4A PROTEASE. AS SUCH, THEY ACT BY INTERFERING WITH THE LIFE CYCLE OF THE HEPATITIS C VIRUS AND ARE ALSO USEFUL AS ANTIVIRAL AGENTS. THE INVENTION FURTHER RELATES TO COMPOSITIONS COMPRISING THESE COMPOUNDS EITHER FOR EX VIVO USE OR FOR ADMINISTRATION TO A PATIENT SUFFERING FROM HCV INFECTION. THE INVENTION ALSO RELATES TO METHODS OF TREATING AN HCV INFECTION IN A PATIENT BY ADMINISTERING A COMPOSITION COMPRISING A COMPOUND OF THIS INVENTION. THE INVENTION FURTHER RELATES TO PROCESSES FOR PREPARING THESE COMPOUNDS.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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