您的位置: 首页 > 农业专利 > 详情页

Aromatic heterocyclic amide compound containing bicyclic nitrogen
专利权人:
Astellas Pharma Inc.
发明人:
OHNUKI, Kei,AZAMI, Hidenori,SAWADA, Yuki,SHIN, Takashi,KURAMOTO, Kazuyuki,KIKUCHI, Shigetoshi,SAITO, Tomoyuki,HAMAGUCHI, Hisao,NAGASHIMA, Takeyuki
申请号:
ES14810281
公开号:
ES2661259T3
申请日:
2014.06.09
申请国别(地区):
ES
年份:
2018
代理人:
摘要:
Compound of the formula (I) or salt thereof: in the formula, R 1 is nitrogen-containing monocyclic aryl or heteroaryl, each of which may be substituted with group (s) selected from the group consisting of halogen, lower alkyl, -O-lower alkyl, halogen-lower alkyl, -O-halogen-lower alkyl, -CN, dimethylamino and cycloalkyl; X is CH, N or C; ** Formula ** is i) a single bond in the case where X is CH or N and ii) a double bond in the case where X is C; Y is a cyclic group described below: ** Formula ** in this case, Y1 is CRh or N, Y2 is CRi or N, provided that Y1 and Y2 are not N at the same time, Ra, Rh and Ri that are equal or different from each other are H or halogen, Rb is H or lower alkyl, Rc is lower alkyl, Y3 is CH or N, Rd and Re which are the same or different from each other are H or lower alkyl, Rf is H or lower alkyl, Y4 is O or S, Y5 is CH or N, Y6 is CH or N, Rg is H or lower alkyl; R2 is H or lower alkyl; R3 and R4 which are the same or different from each other are H, halogen, lower alkyl, -O-lower alkyl, halogen-lower alkyl, -O-halogen-lower alkyl, cycloalkyl, or -CN, or R3 and R4 can form 2 , 2-difluoro-1,3-benzodioxol binding together with the benzene ring to which R3 and R4 are attached; and lower alkyl is a linear or branched alkyl having 1 to 6 carbon atoms.Compuesto de la fórmula (I) o sal del mismo: en la fórmula, R1 es arilo o heteroarilo monocíclico que contiene nitrógeno, cada uno de los cuales puede estar sustituido con grupo(s) seleccionado(s) del grupo que consiste en halógeno, alquilo inferior, -O-alquilo inferior, halógeno-alquilo inferior, -O-halógeno-alquilo inferior, -CN, dimetilamino y cicloalquilo; X es CH, N o C; **Fórmula** es i) un enlace sencillo en el caso en el que X es CH o N y ii) un doble enlace en el caso en el que X es C; Y es un grupo cíclico descrito a continuación:**Fórmula** en este caso, Y1 es CRh o N, Y2 es CRi o N, siempre que Y1 e Y2 no sean N al mismo tiempo, Ra, Rh y Ri que son iguales o diferentes entre sí son
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
相关发明人
相关专利

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充