SÖRGEL, SEBASTIAN,DEFIEBER, CHRISTIAN,LE VEZOUET, RONAN,CULBERTSON, DEBORAH L.,ANSPAUGH, DOUGLAS D.
申请号：
ES11737922
公开号：
ES2531448T3
申请日:
2011.07.18
申请国别(地区):
ES
年份:
2015
代理人:
摘要：
Hetaryl (thio) carboxamide compounds of formula I ** Formula ** in which X is S or O； R1 is C1-C10 alkyl, C1-C10 haloalkyl, C3-C10 alkenyl, C3-C10 alkynyl, C1-C4-CN alkylene, C1-C4-alkylene alkylene, C1-C4 phenyl-alkyl, C3-C10 alkyl-C1-alkyl -C4, saturated 5- or 6-membered heterocyclyl-C1-C4 alkyl, or 5- or 6-membered heteroaryl-C1-C4 alkyl, wherein the cycloalkyl ring and the C3-C10 cycloalkyl heterocyclyl ring-C1- alkyl C4 and heterocyclyl-C1-C4 alkyl, respectively, is unsubstituted or carries 1, 2, 3, 4 or 5 identical or different Ry substituents, and wherein the phenyl ring and the phenyl-C1-alkyl ring C4 and heteroaryl-C1-C4 alkyl, respectively, is unsubstituted or carries 1, 2, 3, 4 or 5 identical or different Ry substituents； A is a 5-membered hetaryl that has the formulas A1, A2, A3, A4, A5, A6, or A7: ** Formula ** in which it represents the point of attachment to the rest of formula I, Z is O, S or N-RN, wherein RN is as defined in claim 1, n is 0, 1, 2, or 3, RA 'is hydrogen, or has one of the meanings given for RA； or is selected from the group consisting of the radicals of formulas A8-1, A8-2, A8-3, A8-4, A8-5, A8-6, A8-7, A8-8, and A8-9: ** Formula ** independently selected from each other from hydrogen, halogen, C1-C4 alkyl, C1-C4 haloalkyl, C1-C4 alkoxy, C1-C4 haloalkoxy, C1-C3-CN alkylene, C1-C3-OR alkylene, C3 cycloalkyl -C7, C3-C7 cycloalkyl-C1-C3 alkyl, heterocyclyl-C1-C3 saturated alkyl of 3 to 7 members, in which cycloalkyl and heterocyclyl in the last 3 radicals mentioned may be unsubstituted or may carry 1, 2, 3 , 4 or 5 identical or different Ry substituents； RA is selected from the group consisting of halogen, CN, NO2, C1-C10 alkyl, C2-C10 alkenyl and C2-C10 alkynyl, in which the last three radicals mentioned may be unsubstituted, may be partially or totally halogenated or they can carry 1, 2 or 3 identical or different Rx substituents, and also between the group consisting of ORa, C (Y) Rb, C (Y) ORc, S (O) mRd, NReRf, heterocyclyl, phenyl
