CHRISTIAN HUBSCHWERLEN,GEORG RUEEDI,CORNELIA ZUMBRUNN ACKLIN,JEAN-PHILIPPE SURIVET
申请号：
MX2014005637
公开号：
MX2014005637A
申请日:
2012.11.07
申请国别(地区):
MX
年份:
2014
代理人:
摘要：
The invention relates to antibacterial compounds of formula I (Fornula I) (I) wherein R1a represents H or carboxy and R1b represents H, or R1a and R1b represent together either the group *-C(0)-NH-S-# or the group *-C(OH)=N-S-# wherein "*" represents the point of attachment of R1a and "#" represents the point of attachment of R1b R2 represents H, (C1-C3)alkyl, hydroxy-(C1C3)alkyl, benzyl or (C3-C5)cycloalkyl R3 represents H or halogen U represents N or CR4 wherein R4 is H or (C1-C3)alkoxy A represents CH, B represents NH and m represents 1 or 2 and n represents 1 or 2 or A represents N, B is absent, m represents 2 and n represents 2 Y represents CH or N and Q represents O or S and salts of such compounds.La invención se refiere a compuestos antibacterianos de la Fórmula 1 (ver Fórmulas) en donde R1a representa H o carboxi y R1b representa H, o R1a y R1b representan juntos el grupo *-C(O)-NH-S-# o el grupo *-C(OH)=N-S-# en donde "*" representa el punto de unión de R1a y "#" representa el punto de unión de R1b R2 representa H, alquilo de 1 a 3 átomos de carbono, hidroxialquilo de 1 a 3 átomos de carbono, bencilo o cicloalquilo de 3 a 5 átomos de carbono R3 representa H o halógeno U representa N o CR4 en donde R4 es H o alcoxi de 1 a 3 átomos de carbono A representa CH, B representa NH y m representa 1 o 2 y n representa 1 o 2 o A representa N, B está ausente, m representa 2 y n representa 2 Y representa CH o N y Q representa O o S y sales de tales compuestos.
