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method of preparing 4- (cyclopropylmethoxy) -n- (3,5-dichloro-1-oxopyridin-4-yl) -5-methoxypyridine-2-carboxamide crystal forms and crystal forms thereof
专利权人:
SANOFI
发明人:
ALEXANDRE GIULIANI,DIDIER BRIGE,HAGIT ELMALEH,MARC-ANTOINE PERRIN,Pascal Billot
申请号:
BR112015011849
公开号:
BR112015011849A2
申请日:
2013.11.28
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
SUMMARY OF THE INVENTION: "Method of preparing 4- (cyclopropylmethoxy) -n- (3,5-dichloro-1-oxopyridin-4-yl) -5-methoxypyridine-2-carboxamide crystal forms" " The present invention relates to a process for preparing 4- (cyclopropylmethoxy) -N- (3,5-dichloro-1-oxopyridin-4-yl) -5-methoxypyridine-2-carboxamide crystal forms of the formula ( i) said crystal forms which are referred to as aaia crystal forms and their use as a medicament. 1/1resumo patente de invenção: "método de preparação de formas de cristal de 4 (ciclopropilmetoxi)-n-(3,5-dicloro-1-oxidopiridin-4-il)-5-metoxipiridina-2-carboxamida e formas de cristal da mesma". a presente invenção refere-se a um processo de preparação de formas de cristal de 4-(ciclopropilmetoxi)-n-(3,5-dicloro-1-oxidopiridin-4-il)-5-metoxipiridina-2-carboxamida de fórmula (i), as referidas formas de cristal, as quais são designadas como formas de cristal a a i a, e sua utilização como um medicamento. 1/1
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