Compounds derived from 4H, 6h 5 oxa - - - - - 2,3,10b triaza benzo [e] azulenes, V1a Receptor Antagonists； extraction process； Pharmaceutical composition that contains it； use in Pathological States such as dysmenorrhea, hypertension, Liver cirrhosis, nephrotic syndrome, anxiety, among others.

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专利权人:

HOFFMANN-LA ROCHE AG.;F

发明人:

DOLENTE, COSIMO,SCHNIDER, PATRICK

申请号：

CL2014000717

公开号：

CL2014000717A1

申请日:

2014.03.24

申请国别(地区):

CL

年份:

2014

代理人:

摘要：

The present invention provides 4H,6H-5-oxa-2,3,10b-triaza-benzo[e]azulenes of the formula wherein R1 and R2 are as defined herein and which act as V1a receptor modulators, and in particular as V1a receptor antagonists, their manufacture, pharmaceutical compositions containing them and their use as medicaments.LA SOLICITUD SE REFIERE ACOMPUESTOS DERIVADOS DE OXI-CICLOHEXIL-4H, 6H-5-OXA-2,3-10B-TRIAZA-BENZO[E]AZULENO, AGONISTA V1A, A UNA COMPOSICIÓN FARMACÉUTICA QUE LOS COMPRENDE, A UN PROCESO DE OBTENCIÓN DE ELLOS Y A SU USO EN EL TRATAMIENTO DE DISMENORREA, DISFUNCIÓN SEXUAL, HIPERTENSIÓN, FALLO CARDIACO, CIRROSIS HEPÁTICA, ENFERMEDADES SNC, ENTRE OTRAS

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