TANOURY GERALD J,NUGENT WILLIAM ALOYSIUS,DVORNIKOVS VADIMS,ROSE PETER JAMISON
申请号:
IN201637015905
公开号:
IN201637015905A
申请日:
2016.05.06
申请国别(地区):
IN
年份:
2016
代理人:
摘要:
A method of preparing Compound (1) or a pharmaceutically acceptable salt thereof: comprises: (a) reacting Compound (X): a pharmaceutically acceptable salt thereof with Compound (Y): in the presence of a palladium catalyst and a carbonate or phosphate base to form compound (Z): or a pharmaceutically acceptable salt thereof and (b) deprotecting the Ts group of Compound (Z) to form Compound (1) or a pharmaceutically acceptable salt thereof.