KOENRAAD JOZEF LODEWIJK MARCEL ANDRIES,ANIL KOUL,JÉRÔME EMILE GEORGES GUILLEMONT,MAGALI MADELEINE SIMONE MOTTE
申请号：
MYPI 20063045
公开号：
MY151030A
申请日:
2006.06.27
申请国别(地区):
MY
年份:
2014
代理人:
摘要：
USE OF A COMPOUND FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF A BACTERIAL INFECTION PROVIDED THAT THE BACTERIAL INFECTION IS OTHER THAN A MYCOBACTERIAL INFECTION, SAID COMPOUND BEING A COMPOUND OF FORMULA (IA) OR (IB) A PHARMACEUTICALLY ACCEPTABLE ACID OR BASE ADDITION SALT THEREOF, A STEREOCHEMICALLY ISOMERIC FORM THEREOF, A TAUTOMERIC FORM THEREOF OR A N-OXIDE FORM THEREOF, WHEREIN R1 IS HYDROGEN, HALO, HALOALKYL, CYANO, HYDROXY, AR, HET, ALKYL, ALKYLOXY, ALKYLTHIO, ALKYLOXYALKYL, ALKYLTHIOALKYL, AR-ALKYL OR DI(AR)ALKYL P IS 1 TO 4 R2 IS HYDROGEN, HYDROXY, MERCAPTO, ALKYLOXY, ALKYLOXYALKYLOXY, ALKYLTHIO, MONO OR DI(ALKYL)AMINO OR WHEREIN Y IS CH2, O, S, NH OR N-ALKYL R3 IS AR OR HET R4 AND R5 EACH INDEPENDENTLY ARE HYDROGEN, ALKYL OR BENZYL OR R4 AND R5 ARE TAKEN TOGETHER INCLUDING THE N TO WHICH THEY ARE ATTACHED R6 IS HYDROGEN, HALO, HALOALKYL, HYDROXY, AR, ALKYL, ALKYLOXY, ALKYLTHIO, ALKYLOXNALKYL, ALKYLTHIOALKYL, AR-ALKYL OR DI(AR)ALKYL OR TWO VICINAL R6 RADICALS MAY BE TAKEN TOGETHER TO FORM -CH=CH-CH=CH- R IS 1 TO 5 R7 IS HYDROGEN, ALKYL, AR OR HET R8 IS HYDROGEN OR ALKYL R9 IS OXO OR R8 AND R9 TOGETHER FORM -CH=CH-N= ALK IS A STRAIGHT OR BRANCHED SATURATED HYDROCARBON RADICAL HAVING FROM 1 TO 6 CARBON ATOMS.
